Remogliflozin etabonate dose | 20 mg | 50 mg | 150 mg | 500 mg | 1000 mg |
---|---|---|---|---|---|
AUC (0–∞) (ng•h/mL) | NQc | 3.70 (46)d | 9.77 (48)d | 36.8 (67)e | 126 (44)f |
AUC (0–t) (ng.h/mL) | 1.61 (67) g | 3.56 (56) | 9.51 (42) | 35.4 (62) | 107 (53) |
C max (ng/mL) | 1.89 (78) | 4.98 (61) | 17.6 (48) | 41.6 (81) | 144 (59) |
T max (h) | 0.625 | 0.625 | 0.515 | 1.25 | 0.625 |
0.33-2.03 | 0.17-1.50 | 0.17-1.50 | 0.33-2.50 | 0.33-2.50 | |
T ½ (h) | NQc | 0.353 (56)d | 0.256 (35)d | 0.263e (27) | 0.707f (56) |