From: Virtual screening and experimental validation of novel histone deacetylase inhibitors
Chemicals | IC50(μM) | |||
---|---|---|---|---|
HepG2 | L02 | MDA-MB-231 | MCF-10A | |
SAHA | 166 ± 9 | 85 ± 2 | 178 ± 13 | 59 ± 10 |
ZINC12555961 | 87 ± 10 | 85 ± 15 | 57 ± 7 | 142 ± 17 |
ZINC02639234 | >200 | >200 | >200 | >200 |
ZINC09715944 | 157 ± 12 | 65 ± 3 | >200 | 47 ± 7 |