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Table 1 Concentration and type of assay used for each experiment

From: Drug-transporter mediated interactions between anthelminthic and antiretroviral drugs across the Caco-2 cell monolayers

 

Concentrations used

Quantification method

 

A

B

Drug

μg/ml

μM

1

PZQ

SQV

PZQ

20

64

HPLC

SQV

20

29.8

2

SQV

PZQ

[3H] SQV

 

1.07

Radiolabeled assay

PZQ

20

64

3

IVM

SQV

[3H] IVM

 

0.01

Radiolabeled assay

SQV

20

29.8

4

SQV

IVM

SQV

20

29.8

HPLC

IVM

20

22.75

5

PZQ

EFV

PZQ

20

64

HPLC

EFV

20

63.4

6

PZQ

NVP

PZQ

20

64

HPLC

NVP

20

75.1

7

IVM

NVP

[3H] IVM

 

0.01

Radiolabeled assay

NVP

20

75.1

8

NVP

IVM

[3H] NVP

 

1.5

Radiolabeled assay

IVM

20

22.75

9

IVM

LPV

[3H] IVM

 

0.02

Radiolabeled assay

LPV

20

31.81

10

LPV

IVM

[3H] LPV

 

1.5

Radiolabeled assay

IVM

20

22.75

11

IVM

EFV

[3H] IVM

 

0.01

Radiolabeled assay

EFV

20

63.34

12

EFV

IVM

[14C] EFV

 

0.01

Radiolabeled assay

IVM

20

22.75

  1. Drug A Drug whose transport is under investigation
  2. Drug B Interacting drug