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Table 2 NMDA receptor binding affinity

From: KEA-1010, a ketamine ester analogue, retains analgesic and sedative potency but is devoid of Psychomimetic effects

Agent IC50
MK-801 7.13 nM
Ketamine 0.7 μM
KEA-1010 134 μM
KEA-1025 313 μM
KEA-1037 2.7 μM