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Table 2 NMDA receptor binding affinity

From: KEA-1010, a ketamine ester analogue, retains analgesic and sedative potency but is devoid of Psychomimetic effects

AgentIC50
MK-8017.13 nM
Ketamine0.7 μM
KEA-1010134 μM
KEA-1025313 μM
KEA-10372.7 μM