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Fig. 6 | BMC Pharmacology and Toxicology

Fig. 6

From: The inhibition of tamoxifen on UGT2B gene expression and enzyme activity in rat liver contribute to the estrogen homeostasis dysregulation

Fig. 6

The inhibition of UGT2B7 activity by tamoxifen in HLMs. A Concentration-dependent inhibition of UGT2B7 activity by tamoxifen in HLMs. B Time-dependent inhibition of UGT2B7 activity by tamoxifen in HLMs. Tamoxifen concentration: , 0 μM; , 6.25 μM; □, 12.5 μM; ■, 25 μM; , 50 μM; ▲, 100 μM. Results are shown as means ± SEM

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