Parameter | Estimate (% RSE)a | bIIV (%RSE) |
---|---|---|
CL/FTT (L/hr) | 7.01 (10) | 70.3 (7) |
CL/FTC (L/hr) | 2.26 (12) | 70.3 (7) |
C/FLCC (L/hr) | 0.539 (24) | 70.3 (7) |
V/F (L/hr) | 150 FIX | Â |
ka (hr −1) | 0.18 FIX |  |
PROP_ERR | 0.12 | Â |
Effect on CL/F TT , CL/F TC and CL/F CC | ||
CYP2B6GG (%) | +93.1 (24%) | Â |
CYP2B6TT (%) | −63.4 (9) |  |
CYP2B6GT (%) | 0 | Â |
10Â kg increase body weight (%) | +21.1 (21) | Â |
Females (%) | +22.2 (67) | Â |